Publications & Works

Publication Network
Journal articles indexed in SCI, SSCI, and AHCI 9

<i>In silico</i> approach reveals <i>N</i>-(5-phenoxythiophen-2-yl)-2-(arylthio)acetamides as promising selective SIRT2 inhibitors: the case of structural optimization of virtual screening-derived hits

GÖZELLE M., BAKAR ATEŞ F., Massarotti A., Ozkan E., Gunindi H. B., ÖZKAN Y., et al.
JOURNAL OF BIOMOLECULAR STRUCTURE & DYNAMICS , vol.43, no.4, pp.1756-1767, 2025 (SCI-Expanded) identifier identifier identifier

2-(Methyl(phenyl)amino)-<i>N</i>-(phenyloxyphenyl)acetamide structural motif representing a framework for selective SIRT2 inhibition

Kaya S. G., Eren G., Massarotti A., Bakar-Ates F., Ozkan E., Gozelle M., et al.
DRUG DEVELOPMENT RESEARCH , vol.85, no.4, 2024 (SCI-Expanded) Sustainable Development identifier identifier identifier

Enzalutamide-human serum albumin interaction: Electrochemical exploration of complex formation and binding parameters

Chenguiti F., Bakirhan N. K., GÖZELLE M., Doulache M., Saidat B., Atici E. B., et al.
Microchemical Journal , vol.201, 2024 (SCI-Expanded) identifier

Hit evaluation results in 5-benzyl-1,3,4-thiadiazole-2-carboxamide based SIRT2-selective inhibitor with improved affinity and selectivity

Gözelle M., Kaya S. G., Aksel A. B., Özkan E., Bakar Ateş F., Özkan Y., et al.
Bioorganic Chemistry , vol.123, pp.105746, 2022 (SCI-Expanded) Sustainable Development identifier identifier identifier

The potential of 4-aryl-6-morpholino-3(2H)-pyridazinone-2-arylpiperazinylacetamide as a new scaffold for SIRT2 inhibition: in silico approach guided by pharmacophore mapping and molecular docking

ŞÜKÜROĞLU M. K., GÖZELLE M., ÖZKAN Y., EREN G.
MEDICINAL CHEMISTRY RESEARCH , vol.30, no.10, pp.1915-1924, 2021 (SCI-Expanded) Creative Commons License Sustainable Development identifier identifier

Hit-to-lead optimization on aryloxybenzamide derivative virtual screening hit against SIRT

Yagci S., Gözelle M., Kaya S. G., Özkan Y., Aksel A. B., Bakar-Ates F., et al.
BIOORGANIC & MEDICINAL CHEMISTRY , vol.30, 2021 (SCI-Expanded) Sustainable Development identifier identifier identifier

Pharmacophore modeling and virtual screening studies to identify novel selective SIRT2 inhibitors

Eren G., Bruno A., Guntekin-Ergun S., Atalay R., Ozgencil F., Özkan Y., et al.
JOURNAL OF MOLECULAR GRAPHICS & MODELLING , vol.89, pp.60-73, 2019 (SCI-Expanded) Sustainable Development identifier identifier identifier

Studies on the synthesis, characterization, cytotoxic activities and plasmid DNA binding of platinum(II) complexes having 2-subsituted benzimidazole ligands

Gözelle M., Kılıç Süloğlu A., Selmanoğlu G., Ramazanoglu N., Açık L., Gumus F.
POLYHEDRON , vol.161, pp.298-308, 2019 (SCI-Expanded) Sustainable Development identifier identifier

Structure-based exploration and pharmacological evaluation of N-substituted piperidin-4-yl-methanamine CXCR4 chemokine receptor antagonists

Adlere I., Sun S., Zarca A., Roumen L., Gözelle M., Viciano C. P., et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY , vol.162, pp.631-649, 2019 (SCI-Expanded) Creative Commons License identifier identifier identifier
Articles Published in Other Journals 3

Linker and tail group modifications on 2-((4-isopropyl-4H-1,2,4-triazol-3-yl)thio)-N-(4-phenoxyphenyl)acetamide to improve SIRT2 inhibitory potency

GÖZELLE M., ÖZKAN Y., EREN G.
FABAD JOURNAL OF PHARMACEUTICAL SCIENCES , vol.49, no.2, pp.317-332, 2024 (Scopus)

Synthesis of 2-Substitutedbenzimidazolium Tetrachloroplatinate(II) Compounds and Their Cytotoxic Activities on Different Cell Lines

Gözelle M., Kılıç Süloğlu A.
FABAD JOURNAL OF PHARMACEUTICAL SCIENCES , vol.47, no.3, pp.281-292, 2022 (Scopus) identifier identifier

Synthesis, Crystal Structure, Spectroscopic and Density Functional Modelling Studies of The 2-Isopropylbenzimidazolium Tetrachloroplatinate(II) Monohydrate

Zeyrek C. T., ÜNVER H., GÖZELLE M., Dilek N., Gumus F.
GAZI UNIVERSITY JOURNAL OF SCIENCE , vol.30, no.1, pp.139-159, 2017 (ESCI) identifier identifier
Papers Presented at Peer-Reviewed Scientific Conferences 12

Design and biological assessment of novel platinum(II) complexes with benzimidazole ligands against cancer cells

GÖZELLE M., GÜLER E. M.
7th International Eurasian Conference on Biological and Chemical Sciences (EurasianBioChem 2024), Turkey, 2 - 04 October 2024, (Summary Text)

Platinum(II) complexes with 2-/3-/4-(benzimidazol-2-yl)phenol: Synthesis, characterization and in vitro cytotoxic activities

GÖZELLE M., ŞİMAY DEMİR Y. D.
6th International Eurasian Conference on Biological and Chemical Sciences (EurasianBioChem 2023), Ankara, Turkey, 11 - 13 October 2023, (Summary Text)

Ariloksi Benzamit Yapısında Sirtuin İnhibitörü Olabilecek Bileşiklerin Tasarımı, Sentezi ve Biyolojik Aktivite Çalışmaları

YAĞCI S., GÖZELLE M., ÖZKAN Y., BAKAR ATEŞ F., EREN G.
VI. Ulusal Farmasötik Kimya Kongresi, İstanbul, Turkey, 26 - 29 August 2022, (Summary Text)

Application of pharmacophore-based virtual screening for novel SIRT6 inhibitors

GÖZELLE M.
4th International Eurasian Conference on Biological and Chemical Sciences (EurasianBioChem 2021), Ankara, Turkey, 24 - 26 November 2021, (Summary Text)

Discovery of 5-Benzyl-1,3,4-oxadiazole/thiadiazole-2-carboxamides as Potential Leads for Selective SIRT2 Inhibition

GÖZELLE M., ÖZKAN Y., EREN G.
GPSS-2021, 3rd International Gazi Pharma Symposium Series, Ankara, Turkey, 8 - 10 September 2021, (Summary Text)

Design and Synthesis of Aryloxy Benzamide Derivatives with Potential Inhibitory Effect against SIRT2

YAGCI S., GÖZELLE M., KAYA S. G., EREN G.
EFMC-YMCS, 6th EFMC Young Medicinal Chemist Symposium, 5 - 06 September 2019, (Summary Text)

2-SÜBSTİTÜE BENZİMİDAZOL TÜREVİ LİGANDLARI TAŞIYAN PLATİN(II) KOMPLEKSLERİNİN SENTEZ VE SİTOTOKSİK ETKİLERİ ÜZERİNDE ÇALIŞMALAR

GÖZELLE M., GÜMÜŞ F., KILIÇ SÜLOĞLU A., SELMANOĞLU G., RAMAZANOĞLU N., AÇIK L.
V. Ulusal Farmasötik Kimya Kongresi, Turkey, 28 April - 01 May 2018, (Summary Text)

Synthesis of Platinum(II) Complexes Containing Optically Active Benzimidazole Ligands

GÖZELLE M., GÜMÜŞ F.
2nd International Gazi Pharma Symposium Series, 11 - 13 October 2017, (Summary Text)

Synthesis, Cytotoxicity and DNA interactions of Platinum(II) Complexes Having Substituted Benzimidazole Ligands

GÖZELLE M., GÜMÜŞ F., KILIÇ SÜLOĞLU A., SELMANOĞLU G., Ramazanoğlu N., AÇIK L.
2nd International Gazi Pharma Symposium Series, 11 - 13 October 2017, (Summary Text)

Synthesis of Platinum(II) Complexes Having 2-Substituted Benzimidazole Ligands

GÖZELLE M., GÜMÜŞ F.
17th Hellenic Symposium on Medicinal Chemistry, 1 - 03 June 2017, (Summary Text)

HOMOLOGY MODELING OF HUMAN NICOTINAMIDE MONONUCLEOTIDE ADENYLYLTRANSFERASE 2 INSIGHTS INTO ISOENZYME SPECIFIC DIFFERENCES USING MOLECULAR DOCKING SIMULATIONS

GÖZELLE M., EREN G.
21st EuroQSAR, Verona, Italy, 4 - 08 September 2016, (Summary Text)

SYNTHESIS CRYSTAL STRUCTURE SPECTROSCOPIC AND DENSITY FUNCTIONAL MODELLING STUDIES OF 2 ISOPROPYLBENZIMIDAZOLIUM TETRACHLOROPLATINATE II MONOHYDRATE

GÖZELLE M., ZEYREK C. T., ÜNVER H., DİLEK N., GÜMÜŞ F.
International Gazi Pharma Symposium Series, 12 - 15 November 2015, (Summary Text)
Books 1

Türk Farmakopesi

TUNÇBİLEK M., YEŞİLADA A., BALKAN A., TOZKOPARAN B., PALASKA E., ÖZKANLI F., et al.
T. C. Sağlık Bakanlığı Türkiye İlaç ve Tıbbi Cihaz Kurumu, Ankara, 2018
Metrics

Publication

25

Publication (WoS)

9

Publication (Scopus)

11

Citation (WoS)

67

H-Index (WoS)

5

Citation (Scopus)

78

H-Index (Scopus)

5

Citation (Scholar)

100

H-Index (Scholar)

5

Project

6

Open Access

2
UN Sustainable Development Goals