Prof.Dr. ERDEN BANOĞLU

SCI, SSCI ve AHCI İndekslerine Giren Dergilerde Yayınlanan Makaleler

A Highly Potent TACC3 Inhibitor as a Novel Anticancer Drug Candidate

Akbulut O., Lengerli D. , Saatci O., Duman E., ŞEKER U. Ö. Ş. , Isik A., et al.

MOLECULAR CANCER THERAPEUTICS, cilt.19, sa.6, ss.1243-1254, 2020 (SCI İndekslerine Giren Dergi)

Encapsulation of the dual FLAP/mPEGS-1 inhibitor BRP-187 into acetalated dextran and PLGA nanoparticles improves its cellular bioactivity

Shkodra-Pula B., Kretzer C., Jordan P. M. , Klemm P., Koeberle A., Pretzel D., et al.

JOURNAL OF NANOBIOTECHNOLOGY, cilt.18, sa.1, 2020 (SCI İndekslerine Giren Dergi)

Discovery of Novel 5-Lipoxygenase-Activating Protein (FLAP) Inhibitors by Exploiting a Multistep Virtual Screening Protocol

OLĞAÇ A. , Carotti A., Kretzer C., Zergiebel S., Seeling A., Garscha U., et al.

JOURNAL OF CHEMICAL INFORMATION AND MODELING, cilt.60, sa.3, ss.1737-1748, 2020 (SCI İndekslerine Giren Dergi)

Evaluation of Cytotoxic Activity of New Benzimidazole-Piperazine Hybrids Against Human MCF-7 and A549 Cancer Cells

ÖZDEMİR A. , Thranli S., ÇALIŞKAN B. , Arka M., BANOĞLU E.

PHARMACEUTICAL CHEMISTRY JOURNAL, cilt.53, sa.11, ss.1036-1046, 2020 (SCI İndekslerine Giren Dergi)

Benzimidazole derivatives as potent and isoform selective tumor-associated carbonic anhydrase IX/XII inhibitors

Uslu A. G. , Maz T. G. , Nocentini A., BANOĞLU E. , Supuran C. T. , ÇALIŞKAN B.

BIOORGANIC CHEMISTRY, cilt.95, 2020 (SCI İndekslerine Giren Dergi)

Protective effect of piceatannol and bioactive stilbene derivatives against hypoxia-induced toxicity in H9c2 cardiomyocytes and structural elucidation as 5-LOX inhibitors

Boccellino M., Donniacuo M., Bruno F., Rinaldi B., Quagliuolo L., Ambruosi M., et al.

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, cilt.180, ss.637-647, 2019 (SCI İndekslerine Giren Dergi)

A Multi-step Virtual Screening Protocol for the Identification of Novel Non-acidic Microsomal Prostaglandin E-2 Synthase-1 (mPGES-1) Inhibitors

Shekfeh S., ÇALIŞKAN B. , Fischer K., Yalcin T., Garscha U., Werz O., et al.

CHEMMEDCHEM, cilt.14, sa.2, ss.273-281, 2019 (SCI İndekslerine Giren Dergi)

Novel Piperazine Amides of Cinnamic Acid Derivatives as Tyrosinase Inhibitors

GÜR MAZ Z. T. , ŞENOL DENİZ F. S. , Shekfeh S., ERDOĞAN ORHAN İ. , BANOĞLU E. , ÇALIŞKAN B.

LETTERS IN DRUG DESIGN & DISCOVERY, cilt.16, sa.1, ss.36-44, 2019 (SCI İndekslerine Giren Dergi)

Optimisation by design of experiment of benzimidazol-2-one synthesis under flow conditions

Mostarda S., Maz T. G. , Piccinno A., Cerra B., BANOĞLU E.

Molecules, cilt.24, sa.13, 2019 (SCI Expanded İndekslerine Giren Dergi)

Synthesis and cellular bioactivities of novel isoxazole derivatives incorporating an arylpiperazine moiety as anticancer agents

ÇALIŞKAN B. , NALBAT E., Ibis K., Guzelcan E. A. , ATALAY R., BANOĞLU E.

JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, cilt.33, sa.1, ss.1352-1361, 2018 (SCI İndekslerine Giren Dergi)

Structural insight into the optimization of ethyl 5-hydroxybenzo[g] indol-3-carboxylates and their bioisosteric analogues as 5-LO/mPGES-1 dual inhibitors able to suppress inflammation

Bruno F., Errico S., Pace S., Nawrozkij M. B. , Mkrtchyan A. S. , Guida F., et al.

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, cilt.155, ss.946-960, 2018 (SCI İndekslerine Giren Dergi)

Drug discovery approaches targeting 5-lipoxygenase-activating protein (FLAP) for inhibition of cellular leukotriene biosynthesis

GÜR MAZ Z. T. , ÇALIŞKAN B. , BANOĞLU E.

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, cilt.153, ss.34-48, 2018 (SCI İndekslerine Giren Dergi)

Identification of multi-target inhibitors of leukotriene and prostaglandin E-2 biosynthesis by structural tuning of the FLAP inhibitor BRP-7

GÜR MAZ Z. T. , ÇALIŞKAN B. , Garscha U., OLĞAÇ A. , Schubert U. S. , Gerstmeier J., et al.

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, cilt.150, ss.876-899, 2018 (SCI İndekslerine Giren Dergi)

Pteryxin - A promising butyrylcholinesterase-inhibiting coumarin derivative from Mutellina purpurea

ERDOĞAN ORHAN İ. , ŞENOL DENİZ F. S. , Shekfeh S., Skalicka-Wozniak K., BANOĞLU E.

FOOD AND CHEMICAL TOXICOLOGY, cilt.109, ss.970-974, 2017 (SCI İndekslerine Giren Dergi)

The potential role of in silico approaches to identify novel bioactive molecules from natural resources

OLĞAÇ A. , ERDOĞAN ORHAN İ. , BANOĞLU E.

FUTURE MEDICINAL CHEMISTRY, cilt.9, sa.14, ss.1663-1684, 2017 (SCI İndekslerine Giren Dergi)

BRP-187: A potent inhibitor of leukotriene biosynthesis that acts through impeding the dynamic 5-lipoxygenase/5-lipoxygenase-activating protein (FLAP) complex assembly

Garscha U., Voelker S., Pace S., Gerstmeier J., Emini B., Liening S., et al.

BIOCHEMICAL PHARMACOLOGY, cilt.119, ss.17-26, 2016 (SCI İndekslerine Giren Dergi)

Synthesis and biological evaluation of C(5)-substituted derivatives of leukotriene biosynthesis inhibitor BRP-7

Levent S., Gerstmeier J., OLĞAÇ A. , Nikels F., Garscha U., Carotti A., et al.

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, cilt.122, ss.510-519, 2016 (SCI İndekslerine Giren Dergi)

4,5-Diarylisoxazol-3-carboxylic acids: A new class of leukotriene biosynthesis inhibitors potentially targeting 5-lipoxygenase-activating protein (FLAP)

BANOĞLU E. , Celikoglu E., Voelker S., OLĞAÇ A. , Gerstmeier J., Garscha U., et al.

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, cilt.113, ss.1-10, 2016 (SCI İndekslerine Giren Dergi)

Crystal structure and DFT calculations of 5-(4-Chlorophenyl)-1-(6-methoxypyridazin-3-yl)-1 H-pyrazole-3-carboxylic acid

ALAŞALVAR C., SOYLU M. S. , ÜNVER H., OCAK İSKELELİ N., YILDIZ M., Ciftci M., et al.

SPECTROCHIMICA ACTA PART A-MOLECULAR AND BIOMOLECULAR SPECTROSCOPY, cilt.132, ss.555-562, 2014 (SCI İndekslerine Giren Dergi)

Synthesis and preliminary mechanistic evaluation of 5-(p-tolyl)-1-(quinolin-2-yl)pyrazole-3-carboxylic acid amides with potent antiproliferative activity on human cancer cell lines

Pirol S. C. , ÇALIŞKAN B. , Durmaz I., ATALAY R., BANOĞLU E.

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, cilt.87, ss.140-149, 2014 (SCI İndekslerine Giren Dergi)

Synthesis, biological evaluation and molecular docking studies of trans-indole-3-acrylamide derivatives, a new class of tubulin polymerization inhibitors

BAYTAŞ S. , Inceler N., Yilmaz A., OLĞAÇ A. , Menevse S., BANOĞLU E. , et al.

BIOORGANIC & MEDICINAL CHEMISTRY, cilt.22, sa.12, ss.3096-3104, 2014 (SCI İndekslerine Giren Dergi)

The novel benzimidazole derivative BRP-7 inhibits leukotriene biosynthesis in vitro and in vivo by targeting 5-lipoxygenase-activating protein (FLAP)

Pergola C., Gerstmeier J., Moench B., Caliskan B. , Luderer S., Weinigel C., et al.

British Journal of Pharmacology, cilt.171, sa.12, ss.3051-3064, 2014 (SCI Expanded İndekslerine Giren Dergi)

Chromatographic separation and biological evaluation of benzimidazole derivative enantiomers as inhibitors of leukotriene biosynthesis

Sardella R., Levent S., Ianni F., ÇALIŞKAN B. , Gerstmeier J., Pergola C., et al.

JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, cilt.89, ss.88-92, 2014 (SCI İndekslerine Giren Dergi)

Pyrazole derivatives as inhibitors of arachidonic acid-induced platelet aggregation

Levent S., ÇALIŞKAN B. , Ciftci M., ÖZKAN Y. , Yenicesu I., ÜNVER H., et al.

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, cilt.64, ss.42-53, 2013 (SCI İndekslerine Giren Dergi)

Synthesis and evaluation of analgesic, anti-inflammatory, and anticancer activities of new pyrazole-3(5)-carboxylic acid derivatives

ÇALIŞKAN B. , Yilmaz A., Evren I., Menevse S., Uludag O. , BANOĞLU E.

MEDICINAL CHEMISTRY RESEARCH, cilt.22, sa.2, ss.782-793, 2013 (SCI İndekslerine Giren Dergi)

Overview of recent drug discovery approaches for new generation leukotriene A(4) hydrolase inhibitors

ÇALIŞKAN B. , BANOĞLU E.

EXPERT OPINION ON DRUG DISCOVERY, cilt.8, sa.1, ss.49-63, 2013 (SCI İndekslerine Giren Dergi)

Identification of novel benzimidazole derivatives as inhibitors of leukotriene biosynthesis by virtual screening targeting 5-lipoxygenase-activating protein (FLAP)

BANOĞLU E. , ÇALIŞKAN B. , Luderer S., EREN G. , Ozkan Y., Altenhofen W., et al.

BIOORGANIC & MEDICINAL CHEMISTRY, cilt.20, sa.12, ss.3728-3741, 2012 (SCI İndekslerine Giren Dergi)

Serum interleukin-16 levels in patients with nasal polyposis

Keseroglu K., BANOĞLU E. , Kizil Y., AYDİL U. , IŞIK GÖNÜL İ. , Yilmaz M. , et al.

Laryngoscope, cilt.122, sa.5, ss.961-964, 2012 (SCI Expanded İndekslerine Giren Dergi)

From Molecular Docking to 3D-Quantitative Structure-Activity Relationships (3D-QSAR): Insights into the Binding Mode of 5-Lipoxygenase Inhibitors

EREN G. , Macchiarulo A., BANOĞLU E.

MOLECULAR INFORMATICS, cilt.31, sa.2, ss.123-134, 2012 (SCI İndekslerine Giren Dergi)

Pyrazol-3-propanoic acid derivatives as novel inhibitors of leukotriene biosynthesis in human neutrophils

ÇALIŞKAN B. , Luderer S., Ozkan Y., Werz O., BANOĞLU E.

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, cilt.46, sa.10, ss.5021-5033, 2011 (SCI İndekslerine Giren Dergi)

Synthesis, antioxidant and antimicrobial evaluation of simple aromatic esters of ferulic acid

Ergun B. , ÇOBAN T., Onurdag F. K. , BANOĞLU E.

Archives of Pharmacal Research, cilt.34, sa.8, ss.1251-1261, 2011 (SCI Expanded İndekslerine Giren Dergi)

Stable ester and amide conjugates of some NSAIDs as analgesic and antiinflammatory compounds with improved biological activity

ULUDAĞ M. O. , Ergun B. , Alkan D. A. , Ercan N., Ozkan G. Y. , BANOĞLU E.

Turkish Journal of Chemistry, cilt.35, sa.3, ss.427-439, 2011 (SCI Expanded İndekslerine Giren Dergi)

Synthesis, biological evaluation, and docking studies of novel heterocyclic diaryl compounds as selective COX-2 inhibitors

EREN G. , Unlu S., Nunez M., Labeaga L., Ledo F., Entrena A., et al.

BIOORGANIC & MEDICINAL CHEMISTRY, cilt.18, sa.17, ss.6367-6376, 2010 (SCI İndekslerine Giren Dergi)

Amide derivatives of [6-acyl-2-benzothiazolinon-3-yl] acetic acids as potential analgesic and anti-inflammatory compounds

ÖNKOL T. , BANOĞLU E. , DÜNDAR Y. , Kupeli E., Sahin M. F.

MEDICINAL CHEMISTRY RESEARCH, cilt.19, sa.1, ss.11-24, 2010 (SCI İndekslerine Giren Dergi)

Carbon Nanotubes to Deliver Drug Molecules

İLBASMIŞ TAMER S. , Yilmaz S., BANOĞLU E. , Degim I. T.

JOURNAL OF BIOMEDICAL NANOTECHNOLOGY, cilt.6, sa.1, ss.20-27, 2010 (SCI İndekslerine Giren Dergi)

Synthesis of 1,5-diarylpyrazol-3-propanoic acids towards inhibition of cyclooxygenase-1/2 activity and 5-lipoxygenase-mediated LTB4 formation

Ergun B. , Teresa Nunez M., Labeaga L., Ledo F., Darlington J., Bain G., et al.

Arzneimittel-Forschung/Drug Research, cilt.60, sa.8, ss.497-505, 2010 (SCI Expanded İndekslerine Giren Dergi)

Synthesis and biological evaluation of 4,5-diphenyloxazolone derivatives on route towards selective COX-2 inhibitors

DÜNDAR Y. , Unlu S., BANOĞLU E. , Entrena A., Costantino G., Nunez M., et al.

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, cilt.44, sa.5, ss.1830-1837, 2009 (SCI İndekslerine Giren Dergi)

Screening and evaluation of antioxidant activity of some pyridazine derivatives

Caliskan-Erguen B. , Suekueroglu M. K. , ÇOBAN T., BANOĞLU E. , SÜZEN S.

JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, cilt.23, sa.2, ss.225-229, 2008 (SCI İndekslerine Giren Dergi)

Synthesis, characterization and preliminary screening of regioisomeric 1-(3-pyridazinyl)-3-arylpyrazole and 1-(3-pyridazinyl)-5-arylpyrazole derivatives towards cyclooxygenase inhibition

Unlu S., BANOĞLU E. , Ito S., Niiya T., EREN G. , Okcelik B., et al.

JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, cilt.22, sa.3, ss.351-361, 2007 (SCI İndekslerine Giren Dergi)

Synthesis of the amide derivatives of 3-[1-(3-pyridazinyl)-5-phenyl-1H-pyrazole-3-yl]propanoic acids as potential analgesic compounds

BANOĞLU E. , Sukuroglu M. K. , Ergun B. , BAYTAŞ S. , Aypar E., Aark M.

TURKISH JOURNAL OF CHEMISTRY, cilt.31, sa.6, ss.677-687, 2007 (SCI İndekslerine Giren Dergi)

Screening and evaluation of rat kidney aldose reductase inhibitory activity of some pyridazine derivatives

Suekueroglu M. K. , Calikan-Erguen B. , Das-Evcimen N., Sarikaya M., BANOĞLU E. , Suzen S.

MEDICINAL CHEMISTRY RESEARCH, cilt.15, ss.443-451, 2007 (SCI İndekslerine Giren Dergi)

Synthesis and analgesic activity of some 4,6-disubstituted-3(2H)-pyridazinone derivatives

Sukuroglu M. K. , Kupeli E., BANOĞLU E. , Unlu S., Yesilada E., Sahin M. F.

ARZNEIMITTELFORSCHUNG-DRUG RESEARCH, cilt.56, sa.5, ss.337-345, 2006 (SCI İndekslerine Giren Dergi)

Synthesis, analgesic, and anti-inflammatory activities of [6-(3,5-dimethyl-4-chloropyrazole-1-yl)-3(2H-pyridazinon-2-yl]acetamides

Sukuroglu M. K. , Ergun B. , Unlu S., Sahin M., Kupeli E., Yesilada E., et al.

ARCHIVES OF PHARMACAL RESEARCH, cilt.28, sa.5, ss.509-517, 2005 (SCI İndekslerine Giren Dergi)

Synthesis of amide derivatives of [6-(3,5-dimethylpyrazol-1-yl)-3(2H)- pyridazinone-2-yl]acetic acid and their analgesic and anti-inflammatory properties

BANOĞLU E. , Akoglu C., Unlu S., Ergun B. , Kupeli E., Yesilada E., et al.

Arzneimittel-Forschung/Drug Research, cilt.55, sa.9, ss.520-527, 2005 (SCI Expanded İndekslerine Giren Dergi)

Amide derivatives of [6-(5-methyl-3-phenylpyrazole-1-yl)-3(2H)pyridazinone-2-yl]acetic acids as potential a analgesic and anti-inflammatory compounds

BANOĞLU E. , Akoglu C., Unlu S., Kupeli E., Yesilada E., Sahin E.

ARCHIV DER PHARMAZIE, cilt.337, sa.1, ss.7-14, 2004 (SCI İndekslerine Giren Dergi)

Investigations of new pyridazinone derivatives for the synthesis of potent analgesic and anti-inflammatory compounds with cyclooxygenase inhibitory activity

Okcelik B., Unlu S., BANOĞLU E. , Kupeli E., Yesilada E., Sahin M.

ARCHIV DER PHARMAZIE, cilt.336, sa.9, ss.406-412, 2003 (SCI İndekslerine Giren Dergi)

Amide derivatives of [5-chloro-6-(2-chloro/fluorobenzoyl)-2-benzoxazolinone-3-yl]acetic acids as potential analgesic and anti-inflammatory compounds

BANOĞLU E. , Okcelik B., Kupeli E., Unlu S., Yesilada E., Amat M., et al.

ARCHIV DER PHARMAZIE, cilt.336, ss.251-257, 2003 (SCI İndekslerine Giren Dergi)

Synthesis of new 4-(5-chloro-2-oxo-3H-benzoxazol-3-yl)butanamide derivatives and their analgesic and anti-inflammatory properties

Gulcan H., Unlu S., BANOĞLU E. , Sahin M., Kupeli E., Yesilada E.

TURKISH JOURNAL OF CHEMISTRY, cilt.27, sa.4, ss.467-476, 2003 (SCI İndekslerine Giren Dergi)

Sulfation of indoxyl by human and rat aryl (phenol) sulfotransferases to form indoxyl sulfate

BANOĞLU E. , King R.

EUROPEAN JOURNAL OF DRUG METABOLISM AND PHARMACOKINETICS, cilt.27, sa.2, ss.135-140, 2002 (SCI İndekslerine Giren Dergi)

Hepatic microsomal metabolism of indole to indoxyl, a precursor of indoxyl sulfate

BANOĞLU E. , Jha G., King R.

EUROPEAN JOURNAL OF DRUG METABOLISM AND PHARMACOKINETICS, cilt.26, sa.4, ss.235-240, 2001 (SCI İndekslerine Giren Dergi)

Simultaneous determination of paracetamol and methocarbamol in tablets by ratio spectra derivative spectrophotometry and LC

Erk N., Ozkan Y., BANOĞLU E. , Ozkan S., Senturk Z.

JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, cilt.24, sa.3, ss.469-475, 2001 (SCI İndekslerine Giren Dergi)

Current status of the cytosolic sulfotransferases in the activation of promutagens and procarcinogens metabolic

BANOĞLU E.

CURRENT DRUG METABOLISM, cilt.1, sa.1, ss.1-30, 2000 (SCI İndekslerine Giren Dergi)

Dissolution tests of benazepril-HCl and hydrochlorothiazide in commercial tablets: comparison of spectroscopic and high performance liquid chromatography methods

BANOĞLU E. , Ozkan Y., Atay O.

FARMACO, cilt.55, ss.477-483, 2000 (SCI İndekslerine Giren Dergi)

Noradrenaline and nitrite-nitrate concentrations in the contralateral testes during ipsilateral spermatic cord torsion is the presence or absence of a testis and epididymis

TANYEL F. C. , Aydin A., BANOĞLU E. , Isimer A., Buyukpamukcu N.

BJU INTERNATIONAL, cilt.83, sa.7, ss.833-836, 1999 (SCI İndekslerine Giren Dergi)

Importance of peri-interactions on the stereospecificity of rat hydroxysteroid sulfotransferase STa with 1-arylethanols

BANOĞLU E. , Duffel M.

CHEMICAL RESEARCH IN TOXICOLOGY, cilt.12, sa.3, ss.278-285, 1999 (SCI İndekslerine Giren Dergi)

alpha-Hydroxytamoxifen is a substrate of hydroxysteroid (alcohol) sulfotransferase, resulting in tamoxifen DNA adducts

Shibutani S., Dasaradhi L., Terashima I., BANOĞLU E. , Duffel M.

CANCER RESEARCH, cilt.58, sa.4, ss.647-653, 1998 (SCI İndekslerine Giren Dergi)

Studies on the interactions of chiral secondary alcohols with rat hydroxysteroid sulfotransferase STa

BANOĞLU E. , Duffel M.

DRUG METABOLISM AND DISPOSITION, cilt.25, sa.11, ss.1304-1310, 1997 (SCI İndekslerine Giren Dergi)

Influence of substrate structure on the catalytic efficiency of hydroxysteroid sulfotransferase STa in the sulfation of alcohols

Chen G., BANOĞLU E. , Duffel M.

CHEMICAL RESEARCH IN TOXICOLOGY, cilt.9, sa.1, ss.67-74, 1996 (SCI İndekslerine Giren Dergi)

Diğer Dergilerde Yayınlanan Makaleler

Crystal structure and Hirshfeld surface analysis of 1-(2,4-dichlorobenzyl)-5-methyl-N-(thiophene-2-sulfonyl)-1H-pyrazole-3-carboxamide

AYDIN A., AKKURT M., GÜR MAZ Z. T. , BANOĞLU E.

ACTA CRYSTALLOGRAPHICA SECTION E-CRYSTALLOGRAPHIC COMMUNICATIONS, cilt.74, ss.747-757, 2018 (ESCI İndekslerine Giren Dergi)

Crystal structure and Hirshfeld surface analysis of methyl 1-(2,4-dichlorobenzyl)-5-methyl-1H-pyrazole-3-carboxylate

AYDIN A., AKKURT M., GÜR MAZ Z. T. , BANOĞLU E.

European Journal of Chemistry, cilt.9, sa.4, ss.347-352, 2018 (Diğer Kurumların Hakemli Dergileri)

Studies on some 2-substituted benzimidazole derivatives and their antimicrobial activity

BANOĞLU E. , Abbasoglu U., ŞAHİN M. G.

Gazi Universitesi Eczacilik Fakultesi Dergisi, cilt.10, sa.1, ss.1-13, 1993 (Diğer Kurumların Hakemli Dergileri)

Hakemli Kongre / Sempozyum Bildiri Kitaplarında Yer Alan Yayınlar

Synthesis of 3,4-Diaryl-5-methylisoxazoles with Potent Antiproliferative Activity Against a Panel of Human Liver and Breast Cancer Cell Lines

LENGERLİ D. , TURANLİ S. , ÇALIŞKAN B. , AKHAN GÜZELCAN E., NALBAT E., ATALAY R., et al.

EFMC-ISMC EFMC-YMCS Virtual Poster Session, 09 Eylül 2020

Vicinal Diaryl Heterocyclic Compounds with Potential Anticancer Activity

TURANLİ S. , ÇALIŞKAN B. , AKHAN GÜZELCAN E., GÜNTEKİN ERGÜN S., ATALAY R., BANOĞLU E.

EFMC-ISMC EFMC-YMCS Virtual Poster Session, 09 Eylül 2020

Synthesis of New Vicinal Diaryl Five-Membered Heterocyclic Compounds with Potential Anticancer Activity

TURANLİ S. , LENGERLİ D. , ÇALIŞKAN B. , AKHAN GÜZELCAN E., NALBAT E., ATALAY R., et al.

8th International Drug Chemistry Conference, 27 Şubat - 01 Mart 2020

DISCOVERY OF NOVEL 5-LIPOXYGENASE ACTIVATING PROTEIN (FLAP) INHIBITORS BY VIRTUAL SCREENING ANDPHARMACOLOGICAL EVALUATION

OLĞAÇ A. , CAROTTI A., Garscha U., Werz O., Macchiarulo A., BANOĞLU E.

22nd European Symposium on Quantitative Structure-Activity RelationshipsTranslational and Health Informatics: Implications for Drug Discovery, 16 - 20 Eylül 2018

EVOLUTION OF SELECTIVE FLAP INHIBITOR BRP-7 INTO MULTI-TARGET INHIBITOR OF FLAP, 5-LO AND MPGES-1 IN THE ARACHIDONIC ACID PATHWAY

GÜR MAZ Z. T. , ÇALIŞKAN B. , OLĞAÇ A. , GERSTMEIER J., GARSCHA U., WERZ O., et al.

EFMC International Symposium on Medicinal Chemistry, Ljubljana, Slovenya, 2 - 06 Eylül 2018, ss.231

SYNTHESIS AND ANTIPROLIFERATIVE EVALUATION OF NOVEL ISOXAZOLE-PIPERAZINE HYBRIDS

ÇALIŞKAN B. , Sinoplu E., İbiş K., AKHAN GÜZELCAN E., ATALAY R., BANOĞLU E.

RICT 2018, 4 - 06 Temmuz 2018

SYNTHESIS, CYTOTOXICITY AND STRUCTURE-ACTIVITYRELATIONSHIPS OF NOVEL ISOXAZOLE DERIVATIVES ASANTICANCER AGENTS

İbiş K., ÇALIŞKAN B. , AKHAN GÜZELCAN E., Sinoplu E., ATALAY R., BANOĞLU E.

RICT 2018, 4 - 06 Temmuz 2018

PROTEIN-LIGAND INTERACTION ANALYSIS THROUGH DOCKING AND MOLECULAR DYNAMIC SIMULATIONS OF KNOWN 5-LIPOXYGENASE-ACTIVATING PROTEIN (FLAP) INHIBITORS

OLĞAÇ A. , CAROTTI A., Macchiarulo A., BANOĞLU E.

RICT 2018 Interfacing Chemical Biology and Drug Discovery 54th International Conference on Medicinal Chemistry, Strasbourg, Fransa, 4 - 06 Temmuz 2018

SANAL TARAMA VE FARMAKOLOJİK DEĞERLENDİRME YOLUYLA YENİ 5-LİPOKSİJENAZ AKTİVE EDİCİ PROTEİN (FLAP) İNHİBİTÖRÜ BİLEŞİKLERİN KEŞFİ

OLĞAÇ A. , CAROTTI A., Garscha U., Werz O., Macchiarulo A., BANOĞLU E.

V. ULUSAL FARMASÖTİK KİMYA KONGRESİ, Erzurum, Türkiye, 28 Nisan - 01 Mayıs 2018

ANTİLÖKOTRİEN ETKİLİ 1,2,5-TRİSÜBSTİTÜEBENZİMİDAZOL TÜREVLERİNİN GELİŞTİRİLMESİ ÜZERİNDE YAPILAN ÇALIŞMALAR

GÜR MAZ Z. T. , ÇALIŞKAN B. , GERSTMEIER J., OLĞAÇ A. , GARSCHA U., WERZ O., et al.

V. ULUSAL FARMASÖTİK KİMYA KONGRESİ, Erzurum, Türkiye, 28 Nisan - 01 Mayıs 2018

Discovery of Tyrosinase Inhibitors from Geranium glaberrimum Boiss. Heldr. Using In Vitro and In Silico Methods

Çelikler Ö., ŞENOL DENİZ F. S. , ÇALIŞKAN B. , GÜR MAZ Z. T. , KAHRAMAN A., ERDOĞAN ORHAN İ. , et al.

The 4th Mediterranean Symposium on Medicinal and Aromatic Plants (MESMAP-2018), 18 - 22 Nisan 2018

Discovery of Novel 5-Lipoxygenase Activating Protein (FLAP) Inhibitors by Virtual Screening

OLĞAÇ A. , CAROTTI A., GERSTMEIER J., GARSCHA U., WERZ O., MACCHIARULO A., et al.

2nd International Gazi Pharma Symposium Series, 11 - 13 Ekim 2017

FROM BATCH TO CONTINUOUS FLOW CHEMISTRY:DOE-ASSISTED OPTIMIZATION OF BENZIMIDAZOL-2-ONESYNTHESIS

GÜR Z. T. , MOSTARDA S., PICCINNO A., ÇALIŞKAN B. , BANOĞLU E. , GIOIELLO A.

2nd International Gazi Pharma Symposium Series, 11 - 13 Ekim 2017

Developing Multi-target Inhibitors of Arachidonic Acid Pathway Based on the FLAP Inhibitor BRP-7

GÜR Z. T. , ÇALIŞKAN B. , GERSTMEIER J., OLĞAÇ A. , GARSCHA U., WERZ O., et al.

2nd International Gazi Pharma Symposium Series, 11 - 13 Ekim 2017

Discovery of Dual FLAP/mPGES-1 Inhibitors for Intervention with Inflammatory Diseases:Medicinal Chemistry Challenges

BANOĞLU E. , ÇALIŞKAN B. , GÜR Z. T. , OLĞAÇ A.

Turkish Japanese Workshop on Bioorganic Medicinal Chemistry Natural Products, 14 Eylül 2017

Tirozinaz İnhibitör Etkili Yeni Sinnamik Asit Türevleri

ÇALIŞKAN B. , GÜR Z. T. , ŞENOL F. S. , SHEKFEH S., ERDOĞAN ORHAN İ. , BANOĞLU E.

29. Ulusal Kimya Kongresi, Türkiye, 10 - 14 Eylül 2017, ss.452

Discovery of Novel Microsomal Prostaglandin E2 Synthase-1 (mPGES-1) Inhibitors Using Structure-Based Virtual Screening.

Shekfeh S., Katrin F., ÇALIŞKAN B. , Garscha U., Werz O., BANOĞLU E.

EFMC-ASMC 2017 International Symposium on Advances in Synthetic and Medicinal Chemistry, 27 - 31 Ağustos 2017

Bioisosteric Tuning of FLAP Inhibitor BRP-7 Towards a More Potent Antiinmlammatory Agent with Multiligand Inhibitor Properties in the Arachidonic Acid (AA) Pathway

GÜR Z. T. , ÇALIŞKAN B. , OLĞAÇ A. , GERSTMEIER J., GARSCHA U., WERZ O., et al.

EFMC-ASMC’xx17 EFMC International Symposium on Advances in Synthetic and Medicinal Chemistry, 27 - 31 Ağustos 2017

Discovery of Novel 5-Lipoxygenase Activating Protein (FLAP) Inhibitors by Combined Ligand- and Structure-Based Virtual Screening

OLĞAÇ A. , CAROTTI A., GERSTMEIER J., GARSCHA U., WERZ O., MACCHIARULO A., et al.

EFMC-ASMC’xx17 EFMC International Symposium on Advances in Synthetic and Medicinal Chemistry, 27 - 31 Ağustos 2017

Araşidonik asit yolağında çoklu ligand (FLAP/5-LO/mPGES-1) özellikte inhibitör etkili BRP-7 türevlerinin geliştirilmesi

BANOĞLU E. , GÜR Z. T. , ÇALIŞKAN B. , GERSTMEIER J., OLĞAÇ A. , GARSCHA U., et al.

1. Anadolu Üniversitesi Eczacılık Sempozyumu, Eskişehir, Türkiye, 1 - 02 Haziran 2017, ss.10

Diarilpirazol Türevi Bileşiğin (BRP-42) Analjezik ve Antienflamatuvar Aktivitesi Üzerinde Çalışmalar

GÖKER G., HAN S. , ÇALIŞKAN B. , BANOĞLU E. , ULUDAĞ M. O.

3rd International Convention of Pharmaceuticals and Pharmacies, İstanbul, Türkiye, 26 - 29 Nisan 2017, ss.752

İzoksazol Türevi Bileşiklerin in-vivo Analjezik ve Antienflamatuvar Aktivitesi Üzerinde Çalışmalar

Örnek Ö., HAN S. , ÇALIŞKAN B. , BANOĞLU E. , ULUDAĞ M. O.

3rd International Convention of Pharmaceuticals and Pharmacies, İstanbul, Türkiye, 26 - 29 Nisan 2017, ss.738

5-Sübstitüe-Benzimidazol Türevi Bileşiğin Farelerde Analjezik ve Antienflamatuvar Aktivite Tarama Çalışması

Göker S., HAN S. , ÇALIŞKAN B. , BANOĞLU E. , ULUDAĞ M. O.

3rd International Convention of Pharmaceuticals and Pharmacies, İstanbul, Türkiye, 26 - 29 Nisan 2017, ss.732

Anticancer activity of novel benzimidazole derivatives against MCF-7 cancer cells

ÖZDEMİR A. , Uzunoglu S., ÇALIŞKAN B. , BANOĞLU E. , ARK M.

Experimental Biology Meeting, Illinois, Amerika Birleşik Devletleri, 22 - 26 Nisan 2017, cilt.31

Structure Guided Design of Novel Isoxazole and Benzimidazole Derivatives as Potent 5 Lipoxygenase 5 LO and 5 LO Activating Protein FLAP Inhibitors

OLĞAÇ A. , CAROTTI A., WERZ O., BANOĞLU E. , MACCHIARULO A.

XXIV National Meeting in Medicinal Chemistry, Perugia, İtalya, 11 - 14 Eylül 2016

Evias Web Services Cloud Based Drug Discovery Platform

OLĞAÇ A. , BUDAK G., OLĞAÇ S. , NUTI R., CAROTTI A., BANOĞLU E.

21st European Symposium on Quantitative Structure-Activity Relationship, Verona, İtalya, 4 - 08 Eylül 2016

Novel BRP 7 Derivatives Targeting FLAP Potent Inhibitors of Leukotriene Biosynthesis

GÜR Z. T. , ÇALIŞKAN B. , GERSTMEIER J., GARSCHA U., OLĞAÇ A. , WERZ O., et al.

3rd EFMC Young Medicinal Chemist Symposium, Manchester, İngiltere, 1 - 02 Eylül 2016

DISCOVERY OF 4 5 DIARYLISOXAZOL 3 CARBOXYLIC ACID SKELETON AS A NOVEL CHEMOTYPE FOR INHIBITION OF 5 LIPOXYGENASE ACTIVATING PROTEIN FLAP

ÇALIŞKAN B. , çelikoğlu e., gerstmeier j., voelker s., garscha u., OLĞAÇ A. , et al.

EFMC International Symposium on Medicinal Chemistry, Manchester, İngiltere, 28 Ağustos - 01 Eylül 2016

Exploratıon of the Chemıcal Space Around C 5 Posıtıon Of The Benzimidazole Nucleus in BRP 7 Towards More Potent Inhıbıtors of Human 5 Lıpoxygenase Actıvatıng Proteın FLAP

GÜR Z. T. , ÇALIŞKAN B. , GERSTMEIER J., OLĞAÇ A. , NIKELS F., WERZ O., et al.

EFMC International Symposium on Medicinal Chemistry 2016, Manchester, İngiltere, 28 Ağustos - 01 Eylül 2016

EXPLORATION OF THE CHEMICAL SPACE AROUND C 5 POSITION OF THE BENZIMIDAZOLE NUCLEUS IN BRP 7 TOWARDS MORE POTENT INHIBITORS OF HUMAN 5 LIPOXYGENASE ACTIVATING PROTEIN FLAP

GÜR Z. T. , ÇALIŞKAN B. , Gerstmeier J., OLĞAÇ A. , nikels F., werz o., et al.

EFMC International Symposium on Medicinal Chemistry, Manchester, İngiltere, 28 Ağustos - 01 Eylül 2016

Discovery of 4 5 Diarylisoxazol 3 Carboxylic Acid Skeleton as a Novel Chemotype for Inhibition of 5 Lipoxygenase Activating Proteın FLAP

ÇALIŞKAN B. , ÇELİKOĞLU E., GERSTMEIER J., VOELKER S., GARSCHA U., OLĞAÇ A. , et al.

EFMC International Symposium on Medicinal Chemistry 2016, Manchester, İngiltere, 28 Ağustos - 01 Eylül 2016

Structure Guided Design of Novel Isoxazole and Benzimidazole Derivatives as Potent FLAP and 5 LO Inhibitors

OLĞAÇ A. , CAROTTI A., BANOĞLU E. , MACCHIARULO A.

IBSS'2016 Resources and Techniques in Computational Drug Discovery, Fas, 23 - 26 Mayıs 2016

Evias Cloud Based Drug Discovery Platform

OLĞAÇ A. , BUDAK G., OLĞAÇ S. , NUTI R., CAROTTI A., BANOĞLU E.

High-Performance Modelling and Simulation for Big Data Applications - Management Committee & Working Group Meeting, Dublin, İrlanda, 25 - 26 Nisan 2016

Structure-Guided Design of Novel Isoxazole and Benzimidazole Derivatives as Potent FLAP and 5-LO Inhibitors: Insights from Molecular Dynamics Simulations

OLĞAÇ A. , CAROTTI A., WERZ O., MACCHIARULO A., BANOĞLU E.

1st International Gazi Pharma Symposium Series, 12 - 15 Kasım 2015

STRUCTURE BASED DESIGN AND SYNTHESIS OF NOVEL BRP 7 DERIVATIVES BEARING C 5 POLAR SUSBTITUENTS AS POTENT FLAP INHIBITORS

GÜR Z. T. , OLĞAÇ A. , Gerstmeiner J., Macchiarulo A., Werz O., ÇALIŞKAN B. , et al.

GPSS 2015, Antalya, Türkiye, 12 - 15 Kasım 2015

İzole Sfenoid Sinüs Cerrahisi 40 vakalık serimiz

ERAVCI F. C. , CEYLAN A. , İLERİ F., USLU S. S. , YILMAZ M. , BANOĞLU E. , et al.

37. ULUSAL KBB BBC KONGRESİ, Türkiye, 28 Ekim - 01 Kasım 2015

Structure-Based Design And Synthesis Of Novel Isoxazole And Benzimidazole Derivatives As Potent FLAP and 5-LO Inhibitors: Insights From Molecular Dynamics Simulations

OLĞAÇ A. , CAROTTI A., WERZ O., BANOĞLU E. , MACCHIARULO A.

Summer School on Drug Design in September in Vienna 2015, Viyana, Avusturya, 20 - 25 Eylül 2015

Structure-Based Design and Synthesis of Novel BRP-7 Derivatives as Potent FLAP Inhibitors: Insights from MolecularDynamics Simulations.

OLĞAÇ A. , GÜR Z. T. , CAROTTI A., ÇALIŞKAN B. , GERSTMEIER J., WERZ O., et al.

EFMC International Symposium on Medicinal Chemistry, LİZBON, Portekiz, 7 - 11 Eylül 2014, ss.162

Towards Pharmacophore and Docking based Virtual Screening of Human P2Y12 Receptor Antagonists with the Homology modeled Protein Structure

EREN G. , BANOĞLU E.

20th EuroQSAR, Understanding Chemical-Biological Interactions, St. Petersburg, Rusya, 31 Ağustos - 04 Eylül 2014

Computer Aided Drug Design Targeting 5LO and FLAP

OLĞAÇ A. , CAROTTI A., WERZ O., MACCHIARULO A., BANOĞLU E.

The First Technical Meeting on High-Throughput Molecular Dynamics 2013, 7 - 08 Kasım 2013

New 4,5-Diarylisoxazole Derivatives as Novel Inhibitors of Human 5-Lipoxygenase (5-LO)

ÇALIŞKAN B. , LUDERER S., GERSTMEIER J., EREN G. , WERZ O., BANOĞLU E.

EFMC-ISMC 2012, XXIInd International Symposium on Medicinal Chemistry, Berlin, Almanya, 2 - 06 Eylül 2012

From Molecular Docking to 3D-Quantitative Structure-Activity Relationships (3D-QSAR): Insights into the Binding Mode of 5-Lipoxygenase Inhibitors

EREN G. , MACCHIARULO A., BANOĞLU E.

EFMC-ISMC 2012, XXIInd International Symposium on Medicinal Chemistry, Berlin, Almanya, 2 - 06 Eylül 2012

New Isoxazole Derivatives as Novel Inhibitors of 5-Lipoxygenase

ÇALIŞKAN B. , LUDERER S., EREN G. , WERZ O., BANOĞLU E.

4th International Symposium on Advanced in Synthetic and Medicinal Chemistry, St. Petersburg, Rusya, 21 - 25 Ağustos 2011

From Molecular Docking to 3D-Quantitative Structure-Activity Relationships (3D-QSAR): Insights into the Binding Mode of 5-Lipoxygenase Inhibitors

EREN G. , MACCHIARULO A., BANOĞLU E.

VIII EWDD, Eighth European Workshop in Drug Design, Siena, İtalya, 22 - 28 Mayıs 2011

An Approach to Combined Ligand- and Structure-Based Virtual Screening and QSAR Studies for Determining Novel 5-Lipoxygenase Inhibitors

EREN G. , BANOĞLU E.

IMMPC-ISPC Joint Meeting, 4th International Meeting on Medicinal and Pharmaceutical Chemistry, 6th International Symposium on Pharmaceutical Chemistry, Ankara, Türkiye, 30 Eylül - 02 Ekim 2010

Studies on Synthesis and In Vitro Cyclooxygenase Inhibitory Activities of Diaryl Heterocyclic Compounds

EREN G. , ÜNLÜ S., NUNEZ M. T. , LABEAGA L., ENTRENA A., BANOĞLU E. , et al.

EFMC-ISMC 2010, XXIst International Symposium on Medicinal Chemistry, Brüksel, Belçika, 5 - 09 Eylül 2010

Combining of Ligand- and Structure-Based Information to Derive a Pharmacophore Model for Determining Novel FLAP Inhibitors

EREN G. , ALTENHOFEN W., BANOĞLU E.

Vienna Summer School on Drug Design, Viyena, Avusturya, 13 - 18 Eylül 2009

Homology Modeling of Human 5-Lipoxygenase and Molecular Docking Simulations of Competitive Inhibitors

EREN G. , ÇALIŞKAN B. , COSTANTINO G., MACCHIARULO A., ÜNLÜ S., ÇAKIR B., et al.

3rd International Meeting on Medicinal and Pharmaceutical Chemistry, IMMPC-3, Antalya, Türkiye, 16 - 21 Ekim 2007

Synthesis of 2-[5,6-diphenyl-3(2H)-pyridazinone-2-yl]acetmide and 3-[5,6-diphenyl-3(2H)-pyridazinone-2-yl]propanamide Derivatives as analgesic and anti-inflammatory agents

DOĞRUER D. S. , ÜNLÜ S., AKKOL E. , BANOĞLU E. , ŞAHİN M. F.

XIXth International Symposium on Medicinal Chemistry, İstanbul, Türkiye, 29 Ağustos - 02 Eylül 2006

Synthesis, Characterizaton and Preliminary Screening of Regioisomeric 1-(3-Pyridazinyl)-3-arylpyrazole and 1-(3-Pyridazinyl)-5-arylpyrazole Derivatives Towards Cyclooxygenase Inhibition

ÜNLÜ S., BANOĞLU E. , SHIGERU I., NIIYA T., EREN G. , ÖKÇELİK B., et al.

XIXth International Symposium on Medicinal Chemistry, ISMC 2006, İstanbul, Türkiye, 29 Ağustos - 02 Eylül 2006

Yayınlar & Eserler

SCI, SSCI ve AHCI İndekslerine Giren Dergilerde Yayınlanan Makaleler

Diğer Dergilerde Yayınlanan Makaleler

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